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Deltorphin II(2-D-Ala), [Tyrosyl-3,5-3H]-, 50µCi (1.85MBq)

Deltorphin II, tritiated at the tyrosyl-3,5 position. Deltorphin II is a selective δ opioid receptor (DOPR) agonist.

For research use only. Not for use in diagnostic procedures

Part number: NET1087050UC
List price: USD 25,720.00
Your price:
USD 25,720.00
USD 25,720.00 /each

Overview

Deltorphin II is a delta opioid receptor agonist. These receptors belong to a group of GPCRs proposed to play a role in analgesia and mood. They are potential drug targets for pain and depression.

We offer both agonist and antagonist radioligands for autoradiographic visualization or performing saturation and competition assays to determine receptor expression levels (Bmax), dissociation constants (Kd), association and dissociation rates (kon and koff), and inhibitor constants (Ki) for a variety of receptors. We develop our radioligands to the highest specific activity possible and provide high purity resulting in low non-specific binding products. Each of our ultra-pure radioligands is fully characterized for pharmacological action and validated in receptor binding assays.

Radiolabeled ligands remain the most sensitive method for probing receptor binding biology; yielding unprecedented sensitivity gives results that technicians and scientists can trust. For over 50 years, Revvity has been a leading supplier of New England Nuclear (NEN) radiochemicals, liquid scintillation cocktails, vials and nuclear counting detection instruments.

References for NET1087:

  1. Heather L. Handl, Josef Vagner, Henry I. Yamamura, Victor J. Hruby, Robert J. Gillies, Development of a lanthanide-based assay for detection of receptor–ligand interactions at the δ-opioid receptor, In Analytical Biochemistry, Volume 343, Issue 2, 2005, Pages 299-307.

Specifications

Molecular Weight
782.9
Application
Drug Discovery & Development
Brand
NEN Radiochemicals
Detection Method
Radiometric
Label Position
Specifically Labeled
One Unit Contains
50.0 µCi
Radionuclide
3H
Radioisotope
H-3
Receptor Type
Opioid
Shipping Conditions
Shipped in Dry Ice
Special Ordering Information
This is a radioactive product - shipping address must have a license to receive radioactive materials.
Therapeutic Area
CNS & Neurologic
Inflammation
Pain
Unit Size
50 µCi

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